主條目:RAAS、Renin-angiotensin-system inhibitor腎素-血管張力素系統抑制劑RASi
可以擴張動脈和靜脈
Renin inhibitor[]
- Aliskiren
- Remikiren
angiotensin-converting enzyme inhibitor(ACEI):降壓主要機轉為減少TPR[]
- captopril
- Enalaprilat用在hypertensive emergency IV
- enalapril(prodrug)→Enalaprilat
- lisinopril
- long-acting、prodrug
- 唯一非腎臟排泄的是fosinopril和moexipril
- benazepril
- perindopril
- quinapril
- ramipril
- trandolapril
angiotensin receptor antagonist[]
- peptide
- saralasin:因為為部份致效劑所以不好
- nonpeptide
- losartan
- valsartan
- candesartan
- olmesartan
- eprosartan
- irbesartan
- telmisartan